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1

[Annual Reports in Medicinal Chemistry] Annual Reports in Medicinal Chemistry Volume 42 Volume 42 || Chapter 17 MAP Kinase Inhibitors in Inflammation and Autoimmune Disorders

Bhagwat, Shripad S.

Année:

2007

Langue:

english

Fichier:

PDF, 156 KB

english, 2007

2

Identification of Druggable Cancer Driver Genes Amplified across TCGA Datasets

Chen, Ying, McGee, Jeremy, Chen, Xianming, Doman, Thompson N., Gong, Xueqian, Zhang, Youyan, Hamm, Nicole, Ma, Xiwen, Higgs, Richard E., Bhagwat, Shripad V., Buchanan, Sean, Peng, Sheng-Bin, Staschke,

Journal:

Année:

2014

Langue:

english

Fichier:

PDF, 3.04 MB

english, 2014

3

Synthesis and Structure—Activity Relationships of 5-Heteroatom-Substituted Pyridopyrimidines as Adenosine Kinase Inhibitors.

Gregory A. Gfesser, Erol K. Bayburt, Marlon Cowart, Stanley DiDomenico, Arthur Gomtsyan, Chih-Hung Lee, Andrew O. Stewart, Michael F. Jarvis, Elizabeth A. Kowaluk, Shripad S. Bhagwat

Journal:

Année:

2003

Fichier:

PDF, 177 KB

2003

4

Synthesis and Biological Evaluation of Pteridine and Pyrazolopyrimidine Based Adenosine Kinase Inhibitors.

Arthur Gomtsyan, Stanley Didomenico, Chih-Hung Lee, Andrew O. Stewart, Shripad S. Bhagwat, Elizabeth A. Kowaluk, Michael F. Jarvis

Journal:

Année:

2004

Fichier:

PDF, 34 KB

2004

5

Synthesis of enantiomerically pure pyrrolidinones as endothelin receptor antagonists

Shripad S. Bhagwat, Candido Gude, Kenneth Chan

Journal:

Tetrahedron Letters

Année:

1996

Langue:

english

Fichier:

PDF, 232 KB

english, 1996

6

α-Mercaptoacyl dipeptides that inhibit angiotensin converting enzyme and neutral endopeptidase 24.11

Shripad S. Bhagwat, Cynthia A. Fink, Candido Gude, Kenneth Chan, Ying Qiao, Yumi Sakane, Carol Berry, Raj D. Ghai

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1995

Langue:

english

Fichier:

PDF, 223 KB

english, 1995

7

3-[6-(2-Dimethylamino-1-imidazol-1-yl-butyl)-naphthalen-2-yloxy]-2,2-dimethyl-propionic acid as a highly potent and selective retinoic acid metabolic blocking agent

Mark J. Mulvihill, Julie L.C. Kan, Andrew Cooke, Shripad Bhagwat, Patricia Beck, Mark Bittner, Cara Cesario, David Keane, Viorica Lazarescu, Anthony Nigro, Christy Nillson, Bijoy Panicker, Vanessa Smi

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2006

Langue:

english

Fichier:

PDF, 125 KB

english, 2006

8

Imidazo[1,5-a]pyrazines: Orally efficacious inhibitors of mTORC1 and mTORC2

Andrew P. Crew, Shripad V. Bhagwat, Hanqing Dong, Mark A. Bittner, Anna Chan, Xin Chen, Heather Coate, Andrew Cooke, Prafulla C. Gokhale, Ayako Honda, Meizhong Jin, Jennifer Kahler, Christine Mantis,

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 1.82 MB

english, 2011

9

N-alkylation of indole ring using Mitsunobu reaction

Shripad S. Bhagwat, Candido Gude

Journal:

Tetrahedron Letters

Année:

1994

Langue:

english

Fichier:

PDF, 280 KB

english, 1994

10

Preparation of the 2,6-dioxa[3.1.1]Bicycloheptane nucleus of thromboxane A2

Shripad S. Bhagwat, Philip R. Hamann, W.Clark Still

Journal:

Tetrahedron Letters

Année:

1985

Langue:

english

Fichier:

PDF, 191 KB

english, 1985

11

Structure–activity studies of 5-substituted pyridopyrimidines as adenosine kinase inhibitors

Marlon Cowart, Chih-Hung Lee, Gregory A. Gfesser, Erol K. Bayburt, Shripad S. Bhagwat, Andrew O. Stewart, Haixia Yu, Kathy L. Kohlhaas, Steve McGaraughty, Carol T. Wismer, Joseph Mikusa, Chang Zhu, Ka

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2001

Langue:

english

Fichier:

PDF, 158 KB

english, 2001

12

Synthesis and biological evaluation of clitocine analogues as adenosine kinase inhibitors

Chih-Hung Lee, Jerome F Daanen, Meiqun Jiang, Haixia Yu, Kathy L Kohlhaas, Karen Alexander, Michael F Jarvis, Elizabeth L Kowaluk, Shripad S Bhagwat

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2001

Langue:

english

Fichier:

PDF, 128 KB

english, 2001

13

N-aryl cinnamides: A novel class of rigid and highly potent leukotriene B4 receptor antagonists

Paul D. Greenspan, Alan J. Main, Shripad S. Bhagwat, Lester I. Barsky, Robert A. Doti, Alan R. Engle, Lisa M. Frey, Huanghai Zhou, Kenneth E. Lipson, Michael H. Chin, Robert H. Jackson, Susan Uziel-Fu

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1997

Langue:

english

Fichier:

PDF, 318 KB

english, 1997

14

Preface: special issue on medicinal chemistry of purines

Kenneth A. Jacobson, Jeff Zablocki, Shripad Bhagwat

Journal:

Purinergic Signalling

Année:

2009

Langue:

english

Fichier:

PDF, 44 KB

english, 2009

15

Kinase inhibitors for the treatment of inflammatory and autoimmune disorders

Shripad S. Bhagwat

Journal:

Purinergic Signalling

Année:

2009

Langue:

english

Fichier:

PDF, 347 KB

english, 2009

16

Lead identification of a potent benzopyranone selective estrogen receptor modulator

Jeffrey A. McKie, Shripad S. Bhagwat, Helen Brady, Mary Doubleday, Leah Gayo, Mathew Hickman, Ravi K. Jalluri, Sak Khammungkhune, Adam Kois, Deborah Mortensen, Normand Richard, John Sapienza, Graziell

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2004

Langue:

english

Fichier:

PDF, 281 KB

english, 2004

17

Synthesis and biological evaluation of 6,7-disubstituted 4-aminopyrido[2,3-d]pyrimidines as adenosine kinase inhibitors

Richard J. Perner, Chih-Hung Lee, Meiqun Jiang, Yu-Gui Gu, Stanley DiDomenico, Erol K. Bayburt, Karen M. Alexander, Kathy L. Kohlhaas, Michael F. Jarvis, Elizabeth L. Kowaluk, Shripad S. Bhagwat

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 210 KB

english, 2005

18

Synthesis and structure-activity relationships of 5-heteroatom-substituted pyridopyrimidines as adenosine kinase inhibitors

Gregory A Gfesser, Erol K Bayburt, Marlon Cowart, Stanley DiDomenico, Arthur Gomtsyan, Chih-Hung Lee, Andrew O Stewart, Michael F Jarvis, Elizabeth A Kowaluk, Shripad S Bhagwat

Journal:

European Journal of Medicinal Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 423 KB

english, 2003

19

4-Substituted proline derivatives that inhibit angiotensin converting enzyme and neutral endopeptidase 24.11.

Shripad S. Bhagwat, Cynthia A. Fink, Candido Gude, Kenneth Chan, Ying Qiao, Yumi Sakane, Carol Berry, Raj D. Ghai

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

1994

Langue:

english

Fichier:

PDF, 271 KB

english, 1994

20

Synthesis and structure of the platelet aggregation factor thromboxane A2

Bhagwat, Shripad S., Hamann, Philip R., Still, W. Clark, Bunting, Stuart, Fitzpatrick, Frank A.

Journal:

Année:

1985

Fichier:

PDF, 339 KB

1985

21

Synthesis and biological evaluation of pteridine and pyrazolopyrimidine based adenosine kinase inhibitors

Arthur Gomtsyan, Stanley Didomenico, Chih-Hung Lee, Andrew O Stewart, Shripad S Bhagwat, Elizabeth A Kowaluk, Michael F Jarvis

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2004

Langue:

english

Fichier:

PDF, 262 KB

english, 2004

22

Constitutive and Inducible Cytochromes P450 in Rat Lung Mitochondria: Xenobiotic Induction, Relative Abundance, and Catalytic Properties

Shripad V. Bhagwat, Jayati Mullick, Haider Raza, Narayan G. Avadhani

Journal:

Toxicology and Applied Pharmacology

Année:

1999

Langue:

english

Fichier:

PDF, 195 KB

english, 1999

23

Flavin-containing monooxygenase mediated metabolism of psychoactive drugs by human brain microsomes

Shubhada Bhamre, Shripad V. Bhagwat, Susarla K. Shankar, Michael R. Boyd, Vijayalakshmi Ravindranath

Journal:

Année:

1995

Langue:

english

Fichier:

PDF, 438 KB

english, 1995

24

Cerebral metabolism of imipramine and a purified flavin-containing monooxygenase from human brain

Shripad V. Bhagwat, Shubhada Bhamre, Michael R. Boyd, Vijayalakshmi Ravindranath

Journal:

Neuropsychopharmacology

Année:

1996

Langue:

english

Fichier:

PDF, 879 KB

english, 1996

25

Novel series of pyrrolotriazine analogs as highly potent pan-Aurora kinase inhibitors

Sunny Abraham, Michael J. Hadd, Lan Tran, Troy Vickers, Janice Sindac, Zdravko V. Milanov, Mark W. Holladay, Shripad S. Bhagwat, Helen Hua, Julia M. Ford Pulido, Merryl D. Cramer, Dana Gitnick, Joyce

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 2.20 MB

english, 2011

26

Preferential effects of nicotine and 4-(N-methyl- N-nitrosamino)-1-(3-pyridyl)-1-butanone on mitochondrial glutathione S-transferase a4-4 induction and increased oxidative stress in the rat brain

Shripad V. Bhagwat, C. Vijayasarathy, Haider Raza, Jayati Mullick, Narayan G. Avadhani

Journal:

Biochemical Pharmacology

Année:

1998

Langue:

english

Fichier:

PDF, 647 KB

english, 1998

27

Multiple forms of cytochrome P450 and associated monooxygenase activities in human brain mitochondria

Shripad V Bhagwat, Michael R Boyd, Vijayalakshmi Ravindranath

Journal:

Biochemical Pharmacology

Année:

2000

Langue:

english

Fichier:

PDF, 590 KB

english, 2000

28

Gene-regulating protein kinases as important anti-inflammatory targets

Shripad S Bhagwat, Anthony M Manning, Merl F Hoekstra, Alan Lewis

Journal:

Drug Discovery Today

Année:

1999

Langue:

english

Fichier:

PDF, 306 KB

english, 1999

29

Further characterization of rat brain flavin-containing monooxygenase: Metabolism of imipramine to its n-oxide

Shripad V. Bhagwat, Shubhada Bhamre, Michael R. Boyd, Vijayalakshmi Ravindranath

Journal:

Biochemical Pharmacology

Année:

1996

Langue:

english

Fichier:

PDF, 923 KB

english, 1996

30

Flavin-containing monooxygenase activity in camel tissues: comparison with rat and human liver enzymes

Haider Raza, Shripad V. Bhagwat, Annie John

Journal:

Comparative Biochemistry and Physiology Part C: Toxicology & Pharmacology

Année:

2004

Langue:

english

Fichier:

PDF, 95 KB

english, 2004

31

Small molecule inhibitors of ganglioside biosynthesis as substrate reduction therapy for the gangliosidoses

Xiaomei Bai, Tram Nguyen, Jillian Brown, Charles Glass, Sergio Duron, Shripad Bhagwat, Brett Crawford

Journal:

Molecular Genetics and Metabolism

Année:

2011

Langue:

english

Fichier:

PDF, 60 KB

english, 2011

32

Small molecule inhibitors of Glycosaminoglycan Biosynthesis as substrate optimization therapy for the Mucopolysaccharidoses

Brett Crawford, Jillian Brown, Kelli Tolmie, Ellen Christie, Jeremy Hanson, Charles Glass, Sergio Duron, Shripad Bhagwat

Journal:

Molecular Genetics and Metabolism

Année:

2011

Langue:

english

Fichier:

PDF, 71 KB

english, 2011

33

Small Molecule Inhibitors of Ganglioside Biosynthesis as Substrate Reduction Therapy for the Gangliosidoses

Xiaomei Bai, Hong Sun, Lan Tang, Jillian R. Brown, Charles A. Glass, Sergio Duron, Shripad S. Bhagwat, Brett E. Crawford

Journal:

Molecular Genetics and Metabolism

Année:

2012

Langue:

english

Fichier:

PDF, 54 KB

english, 2012

34

Catalytic activity and immunohistochemical localization of flavin-containing monooxygenase in rat kidney

Shubhada Bhamre, Susarla K. Shankar, Shripad V. Bhagwat, Vijayalakshmi Ravindranath

Journal:

Année:

1993

Langue:

english

Fichier:

PDF, 783 KB

english, 1993

35

Influence of standard and novel LTB4 analogs on human neutrophil chemotaxis measured by the multiwell cap assay

Stacy Psychoyos, Susan Uziel-Fusi, Shripad Bhagwat, Michael M. Morrissey

Journal:

Journal of Immunological Methods

Année:

1989

Langue:

english

Fichier:

PDF, 504 KB

english, 1989

36

Thromboxane receptor antagonism combined with thromboxane synthase inhibition. 1. (.+-.)-(3-Pyridinylbicycloheptyl)alkanoic acids

Bhagwat, Shripad S., Gude, Candido, Cohen, David S., Lee, Warren, Furness, Patricia, Clarke, Frank H.

Journal:

Journal of Medicinal Chemistry

Année:

1991

Langue:

english

Fichier:

PDF, 2.38 MB

english, 1991

37

Discovery of potent, selective and orally bioavailable imidazo[1,5-a]pyrazine derived ACK1 inhibitors

Jin, Meizhong, Wang, Jing, Kleinberg, Andrew, Kadalbajoo, Mridula, Siu, Kam W., Cooke, Andrew, Bittner, Mark A., Yao, Yan, Thelemann, April, Ji, Qunsheng, Bhagwat, Shripad, Mulvihill, Kristen M., Rech

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2013

Langue:

english

Fichier:

PDF, 1.17 MB

english, 2013

38

Synthesis of thromboxane A2

Bhagwat, Shripad S., Hamann, Philip R., Still, W. Clark

Journal:

Journal of the American Chemical Society

Année:

1985

Langue:

english

Fichier:

PDF, 738 KB

english, 1985

39

Small molecule inhibitors of glycosaminoglycan biosynthesis as substrate optimization therapy for the mucopolysaccharidoses

Brown, Jillian R., Herman, Rob W., Webster, Katherine A., Bhagwat, Shripad S., Crawford, Brett E.

Journal:

Molecular Genetics and Metabolism

Année:

2013

Langue:

english

Fichier:

PDF, 95 KB

english, 2013

40

Novel orally available brain penetrant small molecule inhibitors of ganglioside biosynthesis for the treatment of Sandhoff and Tay–Sachs diseases

Bai, Xiaomei, Sun, Hong, Tang, Lan, Duron, Sergio, Bhagwat, Shripad, Crawford, Brett

Journal:

Molecular Genetics and Metabolism

Année:

2013

Langue:

english

Fichier:

PDF, 309 KB

english, 2013

41

Targeting of NH2-Terminal-Processed Microsomal Protein to Mitochondria: A Novel Pathway for the Biogenesis of Hepatic Mitochondrial P450MT2

Sankar Addya, Hindupur K. Anandatheerthavarada, Gopa Biswas, Shripad V. Bhagwat, Jayati Mullick and Narayan G. Avadhani

Journal:

The Journal of Cell Biology

Année:

1997

Langue:

english

Fichier:

PDF, 1.15 MB

english, 1997

42

Thromboxane receptor antagonism combined with thromboxane synthase inhibition. 3. Pyridinylalkyl-substituted 8-[(arylsulfonyl)amino]octanoic acids

Main, Alan J., Bhagwat, Shripad S., Boswell, Clay, Goldstein, Robert, Gude, Candido, Cohen, David, Furness, Patricia, Lee, Warren, Louzan, Marissa

Journal:

Journal of Medicinal Chemistry

Année:

1992

Langue:

english

Fichier:

PDF, 884 KB

english, 1992

43

Purinergic Approaches in Experimental Therapeutics Edited by Kenneth A. Jacobson and Michael F. Jarvis. Wiley-Liss, New York. 1997. xiv + 581 pp. 16 × 24 cm. ISBN 0-47114071-6. $89.95.

Bhagwat, Shripad S.

Journal:

Journal of Medicinal Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 21 KB

english, 1998

44

Thromboxane receptor antagonism combined with thromboxane synthase inhibition. 4. 8-[[(4-Chlorophenyl)sulfonyl]amino]-4-[3-(3-pyridinyl)propyl]octanoic acid and analogs

Bhagwat, Shripad S., Gude, Candido, Boswell, Clay, Contardo, Nicolina, Cohen, David S., Dotson, Ronald, Mathis, Janice, Lee, Warren, Furness, Patricia, Zoganas, Harry

Journal:

Journal of Medicinal Chemistry

Année:

1992

Langue:

english

Fichier:

PDF, 1.27 MB

english, 1992

45

The P2 Nucleotide Receptors Edited by John T. Turner, Gary A. Weisman, and Jeffrey S. Fedan. Humana Press, Totowa, NJ. 1997. xi + 440 pp. 16 × 23.5 cm. ISBN 0-89603-425-9. $139.00.

Bhagwat, Shripad S.

Journal:

Journal of Medicinal Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 16 KB

english, 1998

46

Preparation of lactone systems. Total synthesis of (.+-.)-quadrone

Bornack, Walter K., Bhagwat, Shripad S., Ponton, John, Helquist, Paul

Journal:

Journal of the American Chemical Society

Année:

1981

Langue:

english

Fichier:

PDF, 251 KB

english, 1981

47

The P2 Nucleotide Receptors Edited by John T. Turner, Gary A. Weisman, and Jeffrey S. Fedan. Humana Press, Totowa, NJ. 1997. xi + 440 pp. 16 × 23.5 cm. ISBN 0-89603-425-9. $139.00.

Bhagwat, Shripad S.

Journal:

Journal of Medicinal Chemistry

Année:

1998

Langue:

english

Fichier:

PDF, 13 KB

english, 1998

48

Thromboxane receptor antagonism combined with thromboxane synthase inhibition. 5. Synthesis and evaluation of enantiomers of 8-[[(4-chlorophenyl)sulfonyl]amino]-4-(3-pyridinylalkyl)octanoic acid

Bhagwat, Shripad S., Gude, Candido, Cohen, David S., Dotson, Ron, Mathis, Janice, Lee, Warren, Furness, Patricia

Journal:

Journal of Medicinal Chemistry

Année:

1993

Langue:

english

Fichier:

PDF, 1.50 MB

english, 1993

49

Crystal Structures of Human Adenosine Kinase Inhibitor Complexes Reveal Two Distinct Binding Modes †

Muchmore, Steven W., Smith, Richard A., Stewart, Andrew O., Cowart, Marlon D., Gomtsyan, Arthur, Matulenko, Mark A., Yu, Haixia, Severin, Jean M., Bhagwat, Shripad S., Lee, Chih-Hung, Kowaluk, Elizabe

Journal:

Journal of Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 655 KB

english, 2006

50

High-Throughput Screening for mTORC1/mTORC2 Kinase Inhibitors Using a Chemiluminescence-Based ELISA Assay

Bhagwat, Shripad V., Kahler, Jennifer, Yao, Yan, Maresca, Paul, Brooks, Maureen, Crew, Andy, Boisclair, Michael, Pachter, Jonathan A.

Journal:

Assay and Drug Development Technologies

Année:

2009

Langue:

english

Fichier:

PDF, 587 KB

english, 2009